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GUC - Drug design - Midterm questions

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GUC Pharmacy: Pharmaceutical Drug Design past exams for midterm

Cover lectures 1-5, their tutorials and all important points (e.g. Ki, deltaG, energy of electrostatic interactions, “four-letters” Schroedinger equation), calculations of deltaG, recognition of drug-receptor interactions, prediction of high- or low-activity ligands based on Craig plot.

Hansch QSAR equations. Explore Molecular Mechanics via Hooke’s Law and Quantum Mechanics through the Schrödinger equation to engineer potent ligands.